Investigation of β-lactam antibacterial drugs, β-lactamases, and penicillin-binding proteins with fluorescence polarization and anisotropy: a review.

نویسنده

  • Adam B Shapiro
چکیده

This review covers the uses of fluorescence polarization and anisotropy for the investigation of bacterial penicillin binding proteins (PBPs), which are the targets of β-lactam antibacterial drugs (penicillins, cephalosporins, carbapenems, and monobactams), and of the β-lactamase enzymes that destroy these drugs and help to render bacterial pathogens resistant to them. Fluorescence polarization and anisotropy-based methods for quantitation of β-lactam drugs are also reviewed. A particular emphasis is on methods for quantitative measurement of the interactions of β-lactams and other inhibitors with PBPs and β-lactamases.

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Investigation of β-lactam antibacterial drugs, β- lactamases, and penicillin-binding proteins with fluorescence polarization and anisotropy: a review

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عنوان ژورنال:
  • Methods and applications in fluorescence

دوره 4 2  شماره 

صفحات  -

تاریخ انتشار 2016